Human ADME-Tox 

The Plexpress Human ADME-tox library provides a simple and flexible way to measure gene expression levels of the CYP (Cytochrome P450) -encoding genes and other relevant tox genes associated with drug metabolism from a single sample. In comparison to RT-qPCR, TRAC (TRanscriptional Analysis with the aid of affinity Capture) will allow quicker, more reliable and cost-efficient measurement of mRNA in hepatocytes or HepaRG cells.

Technical note: Human cytochrome P450 expression screening in primary hepatocytes
 

The Plexpress Human CYP panel offers the followings advantages over alternative methods:

  • Direct measurement from crude cell lysates cultured in 96-well plates
  • No RNA extraction or cDNA conversion required
  • Degradation of RNA avoided, high reproducibility with CVs below 10%
  • Multiple housekeeping genes available for use in the same assay (ACTB, SDHA, B2M, GAPDH, UBC, HPRT, RPL13A)
  • The flexibility of TRAC enables easy customization of the panel and the addition of other genes of interest

For more information please contact us

Human ADME-Tox library